Bisoprolol analogues

Bisoprolol magani ne wanda aka saba wa wa marasa lafiya da cututtuka na zuciya da jijiyoyin jini.

Bayanai don amfani shi ne kamar haka:

Kamar sauran magunguna, bisoprolol na da analogues. Muhimmin sakamako shine m, duk suna rage karfin jini. Amma akwai bambance-bambance tsakanin su.

Me zai iya maye gurbin bisoprolol?

Analogues na miyagun ƙwayoyi Bisoprolol kamar haka:

Bugu da ƙari za mu bincika, a wace bambanci tsakanin magunguna-analogues na Bisoprolol.

Mene ne mafi alhẽri - metoprolol ko bisoprolol?

Metoprolol mai amfani ne mai daraja na bisoprolol. Don haka, alamun da ake amfani dasu suna da yawa. Shin akwai bambanci tsakanin waɗannan kwayoyi? Sai dai itace akwai. Idan aka kwatanta kimar talifarsu ta zamani, wanda zai iya zuwa ga ƙarshe cewa bisoprolol yana da amfani mai yawa, wanda zamu tattauna gaba.

Rabin rabin Bisoprolol shine sa'o'i 10-12, kuma a Metoprolol yana da sa'o'i 3-4. Saboda wannan, bisoprolol za a iya dauka sau ɗaya a rana, yawancin cin abinci na metoprolol yafi girma.

Abinda ke ɗaukar metoprolol zuwa sunadaran plasma shine 88%, yayin da Bisoprolol wannan index ya kai kawai 30%. Kuma fiye da wannan alamar ta ƙasaita, shiri zai fi tasiri. Saboda haka, bisoprolol ya fi tasiri.

Bisoprolol shi ne beta-blocker amphophilic, yana da soluble a cikin ruwa da ƙwayoyi. Sabili da haka, Bisoprolol dan kadan ya shiga cikin shamaki na kwakwalwa da kuma kwakwalwa da hanta. Yayin da kwayar halitta ta cire kawai daga hanta, saboda haka, nauyin da ke kan wannan kwayar zai zama mafi girma.

Carvedilol ko bisoprolol - wanda ya fi kyau?

Carvedilol wani misalin Bisoprolol ne. Kamar metoprolol, carvedilol an ƙarfafa ne kawai a cikin hanta. Saboda haka, a cikin marasa lafiya da cututtukan hanta, za a rage yawan miyagun ƙwayoyi da kuma sashi. Ba kamar Bisoprolol ba, Carvedilol da Metoprolol sun shiga cikin ƙananan kwakwalwa na jini, wanda ya haifar da dama daga illa ta tsakiya.

Bisoprolol ko Egiloc - wanda ya fi kyau?

Kimanin kashi 5 cikin 100 na miyagun ƙwayoyi Egilok suna janye daga jiki tare da fitsari. Sauran an cire ta hanta. Saboda haka, gyaran gyare-gyaren mahimmanci kuma idan akwai matsaloli tare da wannan kwayar. A wasu fannoni, aikin da kwayoyi ya kasance daidai, kuma ɗayan zai iya amincewa da juna.

Sabili da haka, ana iya tabbatar da cewa ayyukan da kwayoyi suke bincika sun kama. Dukansu sun rage karfin jini da kuma zuciya. Amma an gudanar da bincike a cikin An rubuta marasa lafiya a matakin karfin jini a yayin rana. Saboda haka, a sakamakon haka, an gano cewa likitancin Bisoprolol ya ci gaba da tasirinsa a cikin safiya nagari. Wasu analogues ba za su iya yin alfaharin wannan ba. Sun dakatar da su ko kuma rage karfin hawan jini na ragewa aikin sa'o'i 3-4 kafin a dauki nauyin ƙwayar magani.

Har ila yau, binciken ya nuna cewa Bisoprolol yana da kyau wajen sarrafa karfin jini da kuma zuciya a cikin jihohi mai kwantar da hankula da kuma aiki ta jiki. A sakamakon binciken da aka tabbatar da shi, cewa a wannan yanayin Bisoprolol ya fi tasiri, fiye da Metoprolol.