Diclofenac analogues

Diclofenac wani rukuni ne na magungunan da ake amfani da su don cututtuka masu ciwon kumburi na gidajen abinci da tsokoki. Abinda yake aiki na miyagun ƙwayoyi yana nufin magungunan anti-inflammatory masu cututtukan steroidal, waɗanda suke da yawa daga contraindications da sakamako masu illa. A wannan yanayin, sau da yawa akwai buƙatar samun analog - ya fi tasiri kuma a lokaci guda ya ɓace. Har ila yau, ba wanda zai iya nuna cewa masana kimiyya daga Birtaniya sun yi kira don cirewa na Diclofenac saboda, bisa ga karatun su, hakan yana ƙara yawan haɗarin ciwon zuciya , wanda a yau yana daya daga cikin "cututtuka" na 'yan adam. Wannan kira bai da tasiri sosai ga likitoci na gida, kuma Diclofenac har yanzu yana da alaƙa don magani.

Gaba, zamu dubi magunguna da zasu maye gurbin Diclofenac.

Diclofenac Analogs a Injections da Janar Bayani

Ana iya yin amfani da maganganu na diclofenac a cikin injections ba su da wuya a samu, idan kun nema tsarin irin wannan aiki. Diclofenac sodium yana cikin Voltaren, Diklak, Almiral, da sauransu.

Yana da wuya a samu wani wakili irin wannan tare da wani abu mai aiki. Shi ne Arthrosan - babban abu mai amfani - meloxicam. Yana da mai hana zabi na COX-2, wanda shi ma wakili ne na kwayoyin cutar anti-inflammatory marasa steroid, tare da babban bioavailability na 89%. Yana da ban sha'awa cewa Diclofenac, bisa ga umarnin, an yarda a yi amfani dashi a yayin da take ciki, idan amfani ya ba da kanta don la'akari da haɗarin da yaron da mahaifiyarsa, kuma, a lokaci guda, Arthrosan ya saba wa juna a ciki.

Sabili da haka, ana iya cewa Diclofenac wani magani ne na yau da kullum, duk da gargaɗin masana kimiyyar Birtaniya. Arthrosan yana da tasiri mai yawa daga dukkan tsarin jiki.

Analog Diclofenac a cikin ampoules a cikin hanyar meloxicam ba za a yi amfani da dogon lokaci.

Misalin zamani na Diclofenac shine Naproxen. An gabatar da shi a cikin nau'i-nau'i, gels da Allunan, yana da raunin sakamako fiye da diclofenac sodium, amma a daidai wannan lokacin kwayoyi ne mai karfi.

Naproxen yana nufin lokaci guda zuwa 5 kungiyoyi masu maganin magunguna:

Wani magungunan ƙwayar cutar ƙwayar cuta wanda zai maye gurbin Diclofenac shine Ibuprofen. A gaskiya ma, wannan ita ce analog idan muka kwatanta sakamako mai lalacewa, contraindications da alamu. Ibuprofen ya zama abin ƙyama ne na phenylpropionic acid, kuma, kamar sauran NSAIDs, ya hana COX.

Analogues na Diclofenac a cikin Allunan

Analogs na Diclofenac a cikin Allunan, ban da kudi na sama, sune:

Ya kamata a lura cewa Sulindack ba shi da cutarwa ga ciki fiye da Indomethacin, amma a lokaci guda ya fi mai guba ga hanta.

Analogues na diclofenac maganin shafawa

Ƙunƙarar saɓo mafi kyau daga cikin maganganu na Diclofenac shine Clofezon. Phenylbutazone an yarda da shi sosai, amma ya wuce aspirin a sakamakonta. Indomethacin ita ce mafi magungunan maganin magungunan anti-inflammatory mai cututtukan steroidal, kuma an tsara shi a cikin matsanancin hali, yayin da yake haddasa mummunan lalacewa ga jiki.

Diclofenac gel analogues

Mafi kyawun kaddarorin a cikin gels shine Piroxicam da Ketoprofen. Mafi yawan amfani naproxen yana da rauni aiki da ƙananan cutar ga jiki.

Analogues na kyandirori Diclofenac

Indomethacin shine magani mafi mahimmanci ga wannan rukuni, sabili da haka ba'a ba da shawarar yin amfani dashi akai-akai.